Article

Acetamidoglycosylation with Glycal Donors: A One-Pot Glycosidic Coupling with Direct Installation of the Natural C(2)-N-Acetylamino Functionality.

Dipartimento di Chimica Bioorganica Università di Pisa (Italy).
Angewandte Chemie International Edition (Impact Factor: 11.26). 02/2000; 39(1):204-207. DOI: 10.1002/(SICI)1521-3757(20000103)112:13.0.CO;2-U
Source: PubMed

ABSTRACT Nitrogen transfer to glycals: A new method for direct C2-aza-glycosylation with glycal donors has been developed (see scheme), employing the new reagent combination of thianthrene-S-oxide and trifluoroacetic anhydride for glycal activation, in an overall one-pot procedure.

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